Mathias Diebold
M.Sc. Chemie, Doktorand
Institut für Pharmazie und Lebensmittelchemie
Am Hubland, Zimmer e00.001
97074 Würzburg
Tel.: +49 (931) 31-80129
E-Mail: mathias.diebold@siehe_unten
Bitte den Domain Namen in der e-mail Adresse zu uni-wuerzburg.de ändern
Publikationen
“Crystal structure of a covalently linked Aurora-A-MYCN complex”
M. Diebold, L. Schonemann, M. Eilers, C. Sotriffer and H. Schindelin
Acta Cryst. D. 79 (1) (2023) 1-9
DOI: 10.1107/S2059798322011433
"Design, Synthesis, and Evaluation of WD-Repeat-Containing Protein 5 (WDR5) Degraders"
A. Dölle, B. Adhikari, A. Krämer, J. Weckesser, N. Berner, L.-M. Berger, M. Diebold, M. M. Szewczyk, D. Barsyte-Lovejoy, C. H. Arrowsmith, J. Gebel, F. Löhr, V. Dötsch, M. Eilers, S. Heinzlmeir, B. Kuster, C. Sotriffer, E. Wolf and S. Knapp
J. Med. Chem. 64 (15) (2021) 10682-10710
DOI: 10.1021/acs.jmedchem.1c00146
"PROTAC-mediated degradation reveals a non-catalytic function of AURORA-A kinase"
B. Adhikari, J. Bozilovic, M. Diebold, J. D. Schwarz, J. Hofstetter, M. Schröder, M. Wanior, A. Narain, M. Vogt, N. D. Stankovic, A. Baluapuri, L. Schönemann, L. Eing, P. Bhandare, B. Kuster, A. Schlosser, S. Heinzlmeir, C. Sotriffer, S. Knapp, E. Wolf
Nat. Chem. Biol. 16 (2020) 1179-1188
DOI: 10.1038/s41589-020-00652-y
"Autoinhibition Mechanism of the Ubiquitin-Conjugating Enzyme UBE2S by Autoubiquitination"
A. K. L. Liess, A. Kucerova, K. Schweimer, L. Yu, T. I. Roumeliotis, M. Diebold, O. Dybkov, C. Sotriffer, H. Urlaub, J. S. Choudhary, J. Mansfeld, S. Lorenz
Structure 27 (2019) 1195-1210
DOI 10.1016/j.str.2019.05.008